分子視算 堅持卓越
公司首頁 - MSC Home最新消息 - News解決方案 - Solutions產品 - Products服務 - Services支援 - Support關於 - About MSC聯絡我們 - Contact UsEnglish
Eidogen

最新最完整的蛋白質序列、模型、配體、及交互作用之資料庫與搜尋工具。代表產品:TIP, EVE, KKB。Eidogen的蛋白結構資訊整合(TIP: Target Informatics Platform)是世界上第一個整合蛋白結構和知識方法為主的系統。

Eidogen可以節省研究人員的實驗時間,例如給定系統蛋白序列或小分子去檢索,則可以馬上從全世界已發表的所蛋白結構中將相關的結構(包含小分子和蛋白之complex)找出來,並自動演算並疊合結構、小分子、和活性中心。有別於傳統的序列分析,提供研究人員以結構比較的概念來找出符合藥物結合的結構,或者是一系列的蛋白結構。

Eidogen的應用包括:
☆Target Prioritization Applications
 *
Target Druggability Assessment
  ※
Binding Site Property Analysis
       ※Binding Site Selectivity Analysis
       ※
SNP structural mapping and analysis
      
※Drug Resistance Mutation Analysis
       ※
Drug Target Clustering 
    *Animal Model Suitability Analysis 
    *Broad Spectrum Anti-Infective Target Analysis

☆Lead Discovery Applications
  *
Novel Lead Fragment & Scaffold Discovery 
  *Binding Site Property Analysis & HTS Library Selection 
  *
Structure-Based Library Design 
  *VLS Binding Mode Analysis

☆Lead Optimization Applications
  *Structure-Based Ligand Affinity Optimization 
  *Structure-Based Selectivity Optimization 
  *
Structure-Based Broad Spectrum Anti-Infective Optimization 
  *
Structure-Based Co-Inhibitor Affinity Optimization 
  *
"Off-Target" Discovery and Analysis 
  *"Off-Target" Assay Panel Design

☆Opportunity Discovery
   *Novel Drug Rescue Opportunities
      ※Due to Drug-Induced Mutations
      ※Due to Poor Selectivity within a Family
      ※Due to "Off-Target" Interactions 
   
*Novel Drug Redesign Opportunities
   *Novel Drug Binding Site Opportunities
   *Novel Co-Inhibition Opportunities 
   *Novel Anti-infective opportunities

All products from Eidogen-Sertanty, Inc.  
Accelrys - Symyx
ChemAxon
Eidogen
Elsevier
Ingenuity
Integromics
MacVector
Sophia Search
公司首頁 - MSC Home最新消息 - News解決方案 - Solutions產品 - Products服務 - Services支援 - Support關於 - About MSC聯絡我們 - Contact UsEnglish